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/ Products Classification 点击展开+Cat. Number | 10-1298 |
Chemical Name | JNJ-1661010 |
CAS Number | 681136-29-8 |
Mol. Formula | C19H19N5OS |
Mol. Weight | 365.46 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Appearance | Off-white solid |
Application Notes | 98% by TLC NMR (Conforms) |
Synonym | N-Phenyl-4-(3-phenyl-1,2,4-thiadiazol-5-yl)-1-piperazinecarboxamide,4-(3-Phenyl-[1,2,4]thizdiazol-5-yl)-piperazine-1-carboxylic acid phenylamide |
Solubility | Soluble in DMSO (up to 25 mg/ml). |
Storage condition | RT |
Stability | Stable for 2 years as supplied. Solutions in DMSO or ethanol may be stored at -20° for up to 3 months. |
References | JNJ-1661010 (681136-29-8) is a potent and selective FAAH inhibitor. Initially forms a covalent adduct with FAAH but is slowly released, IC50 = 12 nM. 100-fold selectivity for FAAH-1 over FAAH-2. Cell permeable and active in vivo. JNJ-1661010 displays analgesic activity in various animal models.
References/Citations
JNJ-1661010 ,货号10-1298 上海惠诚提供10mg 50mg JNJ-1661010,美国focus原装进口,咨询电话021-60498804 |
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