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/ Products Classification 点击展开+Cat. Number | 282982729338159 |
Chemical Name | CI 988 |
CAS Number | [130332-27-3] |
Mol. Formula | C35H42N4O6 |
Mol. Weight | 614.73 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | 4-[[(1R)-2-[[(2R)-3-(1H-indol-3-yl) -2-methyl-1-oxo-2-[[(tricyclo[3.3.1.13,7]dec-2-ylo xy)carbonyl]amino]propyl]amino]-1-phenylethyl]amin o]-4-oxobutanoic acid |
Solubility | Soluble to 100 mM in DMSO |
Storage condition | Store at +4°C |
References | Potent and selective CCK2 (CCK-B) receptor antagonist that displays ~ 1600-fold selectivity over CCK1 receptors (IC50 values are 1.7 and 2717 nM for CCK2 and CCK1 respectively). Has negligible affinity at a range of other binding sites (IC50 > 10 μM). Exhibits anxiolytic activity following oral administration. Purity: >99 % |