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Cat. Number
282216910897463
Chemical Name
Catestatin
CAS Number
[142211-96-9]
Mol. Formula
C107H173N37O26S
Mol. Weight
2425.84
Qty 1
1mg
Storage condition
Store at -20°C
References

Non-competitive nicotinic cholinergic antagonist; selectively inhibits nicotinic-stimulated catecholamine secretion from chromaffin cells and noradrenergic neurons (IC50 ~ 200 nM). Blocks nicotinic-induced cationic signaling (IC50 ~ 200 - 250 nM) and inhibits nicotinic-agonist induced desensitization of catecholamine release. Also stimulates mast cell release of histamine via a separate mechanism.

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