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/ Products Classification 点击展开+Cat. Number | 281962179923424 |
Chemical Name | AM 251 |
CAS Number | [183232-66-8] |
Mol. Formula | C22H21Cl2IN4O |
Mol. Weight | 555.24 |
Qty 1 |
1mg |
Qty 2 | 50mg |
Synonym | N-(Piperidin-1-yl)-5-(4-iodophenyl) -1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-car boxamide |
Solubility | Soluble to 25 mM in ethanol and to 100 mM in DMSO |
Storage condition | Store at RT |
References |
Potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors. Also potent GPR55 agonist (EC50 = 39 nM). Also available as part of the Cannabinoid CB1 Receptor Tocriset™; and in a fluorescent form (Cat. No. 2540). |
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