服务热线
021-60498804
产品中心
/ Products Classification 点击展开+Cat. Number | Eliprodil |
Chemical Name | Eliprodil |
CAS Number | [119431-25-3] |
Mol. Formula | C20H23ClFNO |
Mol. Weight | 347.86 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | α-(4-Chlorophenyl)-4-[(4-fluoropheny l)methyl]-1-piperidineethanol |
Solubility | Soluble to 25 mM in DMSO |
Storage condition | Desiccate at +4°C |
References | Non-competitive NMDA receptor antagonist that acts at the polyamine modulatory site. Selective for NR2B- over NR2A- and NR2C-containing receptors (IC50 values are 1, > 100 and > 100 μM respectively). Also σ1 ligand (Ki = 0.013 μM). Antagonizes neuronal voltage-gated Ca2+ channels and selectively inhibits the rapid component of the delayed rectifier K+ current (IKr). Neuroprotective. Purity: >98 % |