服务热线
021-60498804
产品中心
/ Products Classification 点击展开+Cat. Number | EHT 1864 |
Chemical Name | EHT 1864 |
CAS Number | [754240-09-0] |
Mol. Formula | C25H27F3N2O4S.2HCl |
Mol. Weight | 581.47 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | 5-(5-(7-(Trifluoromethyl)quinolin-4 -ylthio)pentyloxy)-2-(morpholinomethyl)-4H-pyran-4 -one dihydrochloride |
Solubility | Soluble to 100 mM in water and to 75 mM in DMSO |
Storage condition | Store at +4°C |
References | Inhibitor of Rac family GTPases. Blocks activation by direct binding to Rac1, Rac1b, Rac2 and Rac3 (KD values are 40, 50, 60 and 250 nM respectively). Inhibits Rac, Ras and Tiam-induced growth transformation of NIH-3T3 fibroblasts. Reduces β-amyloid peptide production in vivo. Purity: >98 % |