服务热线
021-60498804
产品中心
/ Products Classification 点击展开+Cat. Number | Thioperamide |
Chemical Name | Thioperamide |
CAS Number | [106243-16-7] |
Mol. Formula | C15H24N4S |
Mol. Weight | 292.44 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | N-Cyclohexyl-4-(imidazol-4-yl)-1-pi peridinecarbothioamide |
Solubility | Soluble to 100 mM in DMSO and to 100 mM in ethanol |
Storage condition | Store at -20°C |
References | Potent histamine H3 and H4 antagonist/inverse agonist. Ki values are 25 and 27 nM for human recombinant H3 and H4 receptors respectively. Blocks eosinophil shape change (IC50 = 1.4 μM) and chemotaxis (IC50 = 519 nM) induced by histamine. Freely crosses the blood-brain barrier. Also available as part of the Histamine H3 Receptor Tocriset™. Purity: >99 % |