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| Cat. Number | Thioperamide |
| Chemical Name | Thioperamide |
| CAS Number | [106243-16-7] |
| Mol. Formula | C15H24N4S |
| Mol. Weight | 292.44 |
| Qty 1 |
10mg |
| Qty 2 | 50mg |
| Synonym | N-Cyclohexyl-4-(imidazol-4-yl)-1-pi peridinecarbothioamide |
| Solubility | Soluble to 100 mM in DMSO and to 100 mM in ethanol |
| Storage condition | Store at -20°C |
| References | Potent histamine H3 and H4 antagonist/inverse agonist. Ki values are 25 and 27 nM for human recombinant H3 and H4 receptors respectively. Blocks eosinophil shape change (IC50 = 1.4 μM) and chemotaxis (IC50 = 519 nM) induced by histamine. Freely crosses the blood-brain barrier. Also available as part of the Histamine H3 Receptor Tocriset™. Purity: >99 % |




