服务热线
021-60498804
产品中心
/ Products Classification 点击展开+Cat. Number | PG 01037 dihydrochloride |
Chemical Name | PG 01037 dihydrochloride |
CAS Number | [790658-27-4] |
Mol. Formula | C26H26Cl2N4O.2HCl |
Mol. Weight | 554.34 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | N-[(2E)-4-[4-(2,3-Dichlorophenyl)-1 -piperazinyl]-2-buten-1-yl]-4-(2-pyridyl)-benzamid e dihydrochloride |
Solubility | Soluble to 100 mM in water and to 100 mM in DMSO |
Storage condition | Desiccate at +4°C |
References | Dopamine D3 receptor antagonist; 133-fold selective for D3 over D2 receptors in vitro (Ki values are 0.70, 93.3 and 375 nM for D3, D2 and D4 receptors respectively). Attenuates abnormal involuntary movements associated with L-DOPA (Cat. No. 3788) in rat models of Parkinson's disease. Inhibits the effects of methamphetamine; attenuates drug-induced behaviors in vivo. Purity: >99 % |
下一个:PG-9 maleate上一个:PG 01 |