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Cat. Number
Ac-RYYRIK-NH2
Chemical Name
Ac-RYYRIK-NH2
CAS Number
[200959-48-4]
Mol. Formula
C44H70N14O9
Mol. Weight
939.12
Qty 1
1mg
Storage condition
Desiccate at -20°C
References
High affinity ligand for the NOP site (Ki = 1.5 nM). Antagonizes nociceptin-stimulated GTP binding in rat brain and the chronotropic effect of nociceptin on rat cardiomyocytes. However, displays potent agonist properties in vivo, inhibiting locomotor activity in mice.
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