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/ Products Classification 点击展开+Cat. Number | Tabimorelin hemifumarate |
Chemical Name | Tabimorelin hemifumarate |
CAS Number | [193079-69-5] |
Mol. Formula | C32H40N4O3.½C4H4O4 |
Mol. Weight | 586.73 |
Qty 1 |
10mg |
Synonym | N-[(2E)-5-Amino-5-methyl-1-oxo-2-he xenyl]-N-methyl-3-(2-naphthalenyl)-D-alanyl-N,Nα-di methyl-D-phenylalaninamide hemifumarate |
Solubility | Soluble to 10 mM in water and to 100 mM in DMSO |
Storage condition | Desiccate at RT |
References | Potent, orally active ghrelin receptor (GHS-R1a) agonist (Ki = 50 nM at human recombinant GHS-R1a). Stimulates GH release from rat pituitary cells with an EC50 value of 2.7 nM. Induces hyperphagia and adiposity in lean rats, but not in leptin signaling-deficient ZDF rats. Purity: >98 % |