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| Cat. Number | T 0156 hydrochloride |
| Chemical Name | T 0156 hydrochloride |
| CAS Number | [324572-92-1] |
| Mol. Formula | C31H29N5O7.HCl |
| Mol. Weight | 620.06 |
| Qty 1 |
10mg |
| Qty 2 | 50mg |
| Synonym | 1,2-Dihydro-2-[(2-methyl-4-pyridiny l)methyl]-1-oxo-8-(2-pyrimidinylmethoxy)-4-(3,4,5- trimethoxyphenyl)-2,7-naphthyridine-3-carboxylic acid methyl ester hydrochloride |
| Solubility | Soluble to 25 mM in ethanol and to 25 mM in DMSO |
| Storage condition | Desiccate at +4°C |
| References | Potent and selective inhibitor of phosphodiesterase type 5 (PDE5); more selective than sildenafil (IC50 values are 0.23, 56 and > 63000 nM for T 0156 and 3.6, 29 and > 270 nM for sildenafil at PDE5, PDE6 and PDEs 1 - 4 respectively). Selective over 30 other enzymes and receptors (IC50 > 10 mM) and potentiates electrical field stimulation-induced relaxation of isolated rabbit corpus cavernosum. Active in vivo. Purity: >99 % |
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