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/ Products Classification 点击展开+Cat. Number | Xanomeline oxalate |
Chemical Name | Xanomeline oxalate |
CAS Number | [141064-23-5] |
Mol. Formula | C14H23N3OS.C2H2O4 |
Mol. Weight | 371.46 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | 3-[4-(Hexyloxy)-1,2,5-thiadiazol-3- yl]-1,2,5,6-tetrahydro-1-methylpyridine oxalate |
Solubility | Soluble to 10 mM in water and to 100 mM in DMSO |
Storage condition | Desiccate at +4°C |
References | Functionally selective muscarinic M1 receptor agonist (EC50 values are 0.3, 5, 42, 52 and 92.5 nM at M1, M3, M5, M4 and M2 receptors respectively). Displays a complex pharmacological profile; reversible and wash-resistant binding resulting in full agonist activity at M1, delayed wash-resistant partial agonist activity at M2 and delayed wash-resistant full agonist activity at M4. Exhibits antipsychotic activity, and improves cognitive deficits and behavioral disturbances in Alzheimer's disease and schizophrenia. Purity: >98 % |