服务热线
021-60498804
| Cat. Number | YM 202074 |
| Chemical Name | YM 202074 |
| CAS Number | [299900-84-8] |
| Mol. Formula | C22H30N4O2S.1.5C4H4O4 |
| Mol. Weight | 588.67 |
| Qty 1 |
10mg |
| Qty 2 | 50mg |
| Synonym | N-Cyclohexyl-6-[[N-(2-methoxyethyl) -N-methylamino]methyl]-N-methylthiazolo[3,2-a]benz oimidazole-2-carboxamide sesquifumarate |
| Solubility | Soluble to 20 mM in water and to 100 mM in DMSO |
| Storage condition | Store at +4°C |
| References | High affinity, selective metabotropic glutamate receptor type 1 (mGlu1) antagonist. Binds an allosteric site of the rat mGlu1 receptor with a Ki of 4.8 nM. Inhibits mGlu1-mediated inositol phosphates production (IC50 = 8.6 nM in rat cerebellar granule cells). Neuroprotective in vivo. Purity: >99 % |
Copyright © 2022 上海惠诚生物科技有限公司
沪ICP备2021037845号-6
